Almitrine dimesylate
CAS No. 29608-49-9
Almitrine dimesylate ( Almitrine mesylate;Almitrine bismesylate;Almitrine bismethanesulfonate )
Catalog No. M20572 CAS No. 29608-49-9
Almitrine dimesylate inhibits selectively the Ca2+-dependent K+ channel and that in rat chemoreceptor cellsused in the treatment of hypoxemic chronic lung diseases.
Purity : >98% (HPLC)
Size | Price / USD | Stock | Quantity |
25MG | 32 | In Stock |
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50MG | 41 | In Stock |
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100MG | 70 | In Stock |
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200MG | 97 | In Stock |
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500MG | Get Quote | In Stock |
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1G | Get Quote | In Stock |
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Biological Information
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Product NameAlmitrine dimesylate
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NoteResearch use only not for human use.
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Brief DescriptionAlmitrine dimesylate inhibits selectively the Ca2+-dependent K+ channel and that in rat chemoreceptor cellsused in the treatment of hypoxemic chronic lung diseases.
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DescriptionAlmitrine dimesylate inhibits selectively the Ca2+-dependent K+ channel and that in rat chemoreceptor cellsused in the treatment of hypoxemic chronic lung diseases.
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SynonymsAlmitrine mesylate;Almitrine bismesylate;Almitrine bismethanesulfonate
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PathwayCell Cycle/DNA Damage
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TargetPotassium Channel
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RecptorPotassium Channel
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Research AreaMetabolic Disease
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Indicationchronic obstructive pulmonary disease
Chemical Information
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CAS Number29608-49-9
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Formula Weight669.76
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Molecular FormulaC28H37F2N7O6S2
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Purity>98% (HPLC)
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SolubilityDMSO:125 mg/mL (186.63 mM)
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SMILESCS(O)(=O)=O.CS(O)(=O)=O.Fc1ccc(cc1)C(N1CCN(CC1)c1nc(NCC=C)nc(NCC=C)n1)c1ccc(F)cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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Retigabine
Retigabine (Ezogabine; D23129) is a Kv7.2-7.5 (KCNQ2-5) neuronal potassium channel opener witrh anticonvulsant activity.
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Tertiapin-Q
A high affinity blocker for inward-rectifier K+ channels, this compound is a stable derivative of the bee venom toxin tertiapin. Binds to ROMK1 (Kir1.1) and GIRK1/4 (Kir3.1/3.4) channels with high affinity (Ki values are 1.3 and 13.3 nM respectively) and is selective over Kir2.1 channels. Derivative tertiapin LQ also available.
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TKIM
TKIM is a TWIK-related potassium channel 1 (TREK-1) inhibitor, binding to the pocket of the intermediate (IM) state of TREK-1.TKIM binds to the pocket of the IM state of TREK-1, which differs from the binding of common inhibitors, which bind to channels in the inactive state.?